Additional file 1 of Significant reduction of activity retention in the kidneys via optimized linker sequences in radiohybrid-based minigastrin analogs
posted on 2024-03-02, 04:42authored byNadine Holzleitner, Sebastian Fischer, Isabel Maniyankerikalam, Roswitha Beck, Constantin Lapa, Hans-Jürgen Wester, Thomas Günther
Additional file 1. Characterization of all CCK-2R-targeted compounds (Figure S1-S12) evaluated in this work, as well as additional information on the synthesis of the SiFA-ipa building block, labeling procedures, in vitro experiments, as well as CCK-2R affinity, lipophilicity, and human serum albumin binding data (Table S1), biodistribution data (Table S2) and tumor-to-background ratios (Table S3).
Funding
Deutsche Forschungsgemeinschaft Technische Universität München (1025)