Figure_4.tif (252.11 kB)
Chart 1.
figure
posted on 2012-11-21, 02:21 authored by Peter Kolb, Khai Phan, Zhan-Guo Gao, Adam C. Marko, Andrej Sali, Kenneth A. JacobsonReference compounds (known selective A1AR antagonists) mentioned in the text. Ki values are as follows, with targets other than human A1AR in parentheses: 1: Ki 0.8 nM [8]; 2: Ki 18 nM; 3: Ki 1 nM; 4: Ki 1 nM [11]; 5: Ki 3 nM (bovine A1AR [20]); 6: Ki 584 nM [21].
