Selective Phosphoramidation and Phosphonation of Benzoxazoles
via Sequence Control
Posted on 2017-04-21 - 12:34
A selective
phosphoramidation and phosphonation of benzoxazole
was developed with trialkyl phosphites in the presence of iodine under
mild conditions. In the reaction, the transformation completes in
10 min at room temperature and the substrates are well tolerant, as
2-substituted azoles could afford the quaternary carbon-centered products.
Significantly, phosphites could be selectively introduced into the
C- and N-positions of the benzoxazoles by controlling the addition
sequence and the ratio of substrates.
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Huang, Ling; Gong, Jiuhan; Zhu, Zheng; Wang, Yufeng; Guo, Shengmei; Cai, Hu (2017). Selective Phosphoramidation and Phosphonation of Benzoxazoles
via Sequence Control. ACS Publications. Collection. https://doi.org/10.1021/acs.orglett.7b00726
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AUTHORS (6)
LH
Ling Huang
JG
Jiuhan Gong
ZZ
Zheng Zhu
YW
Yufeng Wang
SG
Shengmei Guo
HC
Hu Cai