Copper-Catalyzed Regioselective sp<sup>3</sup> C–H Azidation of Alkyl Substituents of Indoles and Tetrahydrocarbazoles

Published on 2019-09-11T14:46:36Z (GMT) by
An efficient regioselective sp<sup>3</sup> C–H azidation is developed using CuBr as the catalyst and Zhdankin azidoiodinane as the “N<sub>3</sub>” source. Under simple and mild reaction conditions, the azido group could be successfully incorporated into the sp<sup>3</sup> C–H alkyl substituents of indoles and tetrahydrocarbazoles.

Cite this collection

Huang, Liwu; Xun, Xudong; Zhao, Man; Xue, Jianzhong; Li, Guofeng; Hong, Liang (2019): Copper-Catalyzed Regioselective

sp3 C–H

Azidation of Alkyl Substituents of Indoles and Tetrahydrocarbazoles. ACS Publications. Collection.