Construction of Azepino[2,3‑b]indole Core via Sulfur Ylide
Mediated Annulations

Li, Qing-Zhu

Construction of Azepino[2,3‑b]indole Core via Sulfur Ylide Mediated Annulations

Posted on 2018-11-16 - 19:39

A novel [4 + 3] annulation of indoline-based aza-dienes and crotonate-derived sulfur ylides is described. This method could be further expanded by using more efficient synthetic strategies, including three-component [3 + 1 + 3] cascade and the direct sulfide-catalyzed [4 + 3] cyclization. These protocols enable the rapid construction of azepino[2,3-b]indole cores, and a broad spectrum of the desired products with diverse substituents was facilely accessed in generally high yield.

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Li, Jun-Long; Dai, Qing-Song; Yang, Kai-Chuan; Liu, Yue; Zhang, Xiang; Leng, Hai-Jun; et al. (2018). Construction of Azepino[2,3‑b]indole Core via Sulfur Ylide Mediated Annulations. ACS Publications. Collection. https://doi.org/10.1021/acs.orglett.8b03363

https://doi.org/10.1021/acs.orglett.8b03363

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