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Download fileAntimycobacterial activities and in vitro ADME profiles of wollamide B (1c).
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posted on 2017-04-19, 17:51 authored by Henok Asfaw, Katja Laqua, Anna Maria Walkowska, Fraser Cunningham, Maria Santos Martinez-Martinez, Juan Carlos Cuevas-Zurita, Lluís Ballell-Pages, Peter ImmingAntimycobacterial activities and in vitro ADME profiles of wollamide B (1c).
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MICstabilitywollamide BanalogueTB agent Wollamide BSARADMEcationic antimycobacterial cyclohexapeptideMycobacteriumbovi3.1H 37Rv Parallely1.1 μ M100 μ Mantimycobacterial activity vscompounds 7 cHepG 2 cellsphase peptide synthesis approachstructure-activity relationship studypharmacokinetic propertiesIC