Palladium-Catalyzed Ring-Opening
Reaction of Methyleneaziridines with
Carboxylic Acids:  Synthesis of
α-Amidoketones

Oh, Byoung Ho; Nakamura, Itaru; Yamamoto, Yoshinori

doi:10.1021/jo035739g.s001

jo035739g_si_001.pdf (298.22 kB)

Palladium-Catalyzed Ring-Opening Reaction of Methyleneaziridines with Carboxylic Acids: Synthesis of α-Amidoketones

journal contribution

posted on 2004-04-16, 00:00 authored by Byoung Ho Oh, Itaru Nakamura, Yoshinori Yamamoto

In the presence of palladium catalysts, the reaction of methyleneaziridines 1 with carboxylic acids 2 proceeded smoothly to give the corresponding α-amidoketones 3 in good to high yields.

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Keywords

presence Methyleneaziridine carboxylic acids 2 Synthesi palladium catalysts Amidoketone Acid amidoketone Carboxylic yield methyleneaziridines 1

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